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Scoulerine
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-20°C, sealed storage, away from moisture and light
(-)-Scoulerine; Discretamine
货期:1-2天
MedChemExpress LLC
6451-73-6
1 mg
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CAS No. : 6451-73-6
MCE 国际站:Scoulerine
产品活性:Scoulerine ((-)-Scoulerine) 是一种有效的抗有丝分裂 (antimitotic) 化合物。Scoulerine 也是 BACE1 (淀粉样前体蛋白裂解酶 1) 的抑制剂。Scoulerine 抑制细胞增殖,阻止细胞周期,并诱导癌细胞凋亡。
研究领域:Cell Cycle/DNA Damage | Cytoskeleton | Neuronal Signaling | Apoptosis
作用靶点:Microtubule/Tubulin | Beta-secretase | Apoptosis
In Vitro: Scoulerine ((-)-Scoulerine) inhibits mini-panel of human leukemic cells, MOLT-4 (WT), Jurkat (TP53 mutated), Raji (TP53 mutated), HL-60 (TP53 null), U-937 (TP53 mutated), and HEL 92.1.7 (wild-type), with IC50s ranging from 2.7 µM to 6.5 µM.Scoulerine (2.5-20 µM; 24 hours) decreases proliferation of Jurkat and MOLT-4 cells.Scoulerine (2.5-20 µM; 24 hours) induces MOLT-4 and Jurkat cells apoptosis.Scoulerine induces G2 or M cell cycle arrest.Scoulerine (2.5-5 µM; 24 hours) shows an upregulation of p53 protein in p53 wild-type MOLT-4 cells.Scoulerine (2.5-5 µM; 24-48 hours) activates caspase-3/7, -8 and -9 in a dose-dependent manner.Scoulerine (5-10 µM; 24 hours) disrupts microtubule structure of A549 lung carcinoma cells
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