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- 详细信息
- 技术资料
- 保存条件:
-20°C, sealed storage, away from moisture
- 英文名:
R 24571
- 库存:
货期:1-2天
- 供应商:
MedChemExpress LLC
- CAS号:
57265-65-3
- 规格:
10 mM * 1 mL/1 mg/5 mg/10 mg/25 mg/50 mg/100 mg/200 mg
| 规格: | 10 mM * 1 mL | 产品价格: | ¥983.0 |
|---|---|---|---|
| 规格: | 1 mg | 产品价格: | ¥295.0 |
| 规格: | 5 mg | 产品价格: | ¥650.0 |
| 规格: | 10 mg | 产品价格: | ¥1000.0 |
| 规格: | 25 mg | 产品价格: | ¥1608.0 |
| 规格: | 50 mg | 产品价格: | ¥2413.0 |
| 规格: | 100 mg | 产品价格: | ¥3378.0 |
| 规格: | 200 mg | 产品价格: | ¥4963.0 |
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Calmidazolium chloride
CAS No. : 57265-65-3
MCE 国际站:Calmidazolium chloride
产品活性:Calmidazolium chloride (R 24571) 是一种钙调蛋白拮抗剂,拮抗CaM依赖性磷酸二酯酶和钙调蛋白诱导的红细胞Ca2+转运ATP酶活化, IC50 分别为0.15和0.35 μM。也用于抗癌研究。它结合CaMK的Kd 值为3 nM。
研究领域:Autophagy | Membrane Transporter/Ion Channel
作用靶点:Autophagy | Calmodulin
In Vitro: Calmidazolium chloride is widely used as a calmodulin (CaM) antagonist, but is also known to induce apoptosis in certain cancer cell lines. Calmidazolium chloride (3, 5, 7, 10 μM, 30 minutes-24 hours) inhibits growth of mouse F9 ECCs.
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