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- 详细信息
- 技术资料
- 保存条件:
4°C, sealed storage, away from moisture
- 英文名:
SR57746A; SR57746 hydrochloride
- 库存:
货期:1-2天
- 供应商:
MedChemExpress LLC
- CAS号:
90494-79-4
- 规格:
10 mM * 1 mL/1 mg/5 mg/10 mg/25 mg/50 mg
| 规格: | 10 mM * 1 mL | 产品价格: | ¥873.0 |
|---|---|---|---|
| 规格: | 1 mg | 产品价格: | ¥411.0 |
| 规格: | 5 mg | 产品价格: | ¥950.0 |
| 规格: | 10 mg | 产品价格: | ¥1500.0 |
| 规格: | 25 mg | 产品价格: | ¥3000.0 |
| 规格: | 50 mg | 产品价格: | ¥4600.0 |
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Xaliproden hydrochloride
CAS No. : 90494-79-4
MCE 国际站:Xaliproden hydrochloride
产品活性:Xaliproden hydrochloride (SR57746A) 是一种有效、选择性和具有口服活性的 5-HT1A 受体激动剂,对大鼠海马中的 5-HT1A 特异性结合位点表现出高亲和力 (IC50=3 nM)。Xaliproden hydrochloride 也是一种选择性的多巴胺 D2 受体拮抗剂,具有中等亲和力 (IC50=0.1-1 μM)。Xaliproden hydrochloride 具有抗抑郁作用和抗焦虑作用,并且具有研究神经退行性疾病的潜力。
研究领域:GPCR/G Protein | Neuronal Signaling
作用靶点:5-HT Receptor | Dopamine Receptor
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