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- 2025年12月05日
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- 文献和实验
- 技术资料
- 保存条件：
Please store the product under the recommended conditions in the Certificate of Analysis.
- 英文名：
CB1 inverse agonist 1
- 库存：
货期：询盘
- 供应商：
MedChemExpress LLC
- CAS号：
852315-00-5
- 规格：
1 mg
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MRL-650
CAS No. : 852315-00-5
MCE 国际站：MRL-650
产品活性：MRL-650 (CB1 inverse agonist 1) 是一种高效的，具有口服活性的，特异性 CB1 受体的反向激动剂，对 CB1 和 CB2 受体的 IC50 分别为 7.5 nM 和 4100 nM。具有抑制食欲作用。
研究领域：GPCR/G Protein | Neuronal Signaling
作用靶点：Cannabinoid Receptor
In Vivo: MRL-650 (Compound 14; 0.3, 1, or 3 mg/kg）inhibits feeding in a dose-dependent manner.
The pharmacokinetic profile of CB1 inverse agonist 1 is evaluated in Sprague-Dawley rats, C57BL/6 mice, beagles, and rhesus macaques with t1/2 of >8, >8, >24, and 22 h, respectively.
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文献和实验-2 Digitonin 235 1,229 70,000 - - C12 E8 - 542 65,000 0.005 8.7 x 10-5 Lubrol PX - 582 64,000 0.006 1.0 x 10-4 Triton X-100 - 650 90,000 0.021 3.0 x 10-4 Nonident P-40 - 603 90,000 0.017 3.0 x 10-4 Tween 80
Yeast Nuclear Extract (Small Scale)
Yeast Nuclear Extract (Small Scale) Hahn Lab (adapted from J. Leatherwood, Ptashne lab) last modified Mon, Aug 27, 2001 Cell Growth 3 liters of cells are grown in YPD (3% glucose) to A600 of 3-5. Antifoam A (two drops
Yeast Nuclear Extract (Small Scale)
Hahn Lab (adapted from J.Leatherwood,Ptashne lab) last modified Mon,Aug 27,2001 Cell Growth 3 liters of cells are grown in YPD (3% glucose)to A600 of 3-5.Antifoam A (two drops from a P200 pipetman)is added to media before autoclaving. For wild
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