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- 2025年12月05日
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- 文献和实验
- 技术资料
- 保存条件：
Please store the product under the recommended conditions in the Certificate of Analysis.
- 英文名：
CB1 inverse agonist 1
- 库存：
货期：询盘
- 供应商：
MedChemExpress LLC
- CAS号：
852315-00-5
- 规格：
1 mg
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MRL-650
CAS No. : 852315-00-5
MCE 国际站：MRL-650
产品活性：MRL-650 (CB1 inverse agonist 1) 是一种高效的，具有口服活性的，特异性 CB1 受体的反向激动剂，对 CB1 和 CB2 受体的 IC50 分别为 7.5 nM 和 4100 nM。具有抑制食欲作用。
研究领域：GPCR/G Protein | Neuronal Signaling
作用靶点：Cannabinoid Receptor
In Vivo: MRL-650 (Compound 14; 0.3, 1, or 3 mg/kg）inhibits feeding in a dose-dependent manner.
The pharmacokinetic profile of CB1 inverse agonist 1 is evaluated in Sprague-Dawley rats, C57BL/6 mice, beagles, and rhesus macaques with t1/2 of >8, >8, >24, and 22 h, respectively.
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文献和实验-2 Digitonin 235 1,229 70,000 - - C12 E8 - 542 65,000 0.005 8.7 x 10-5 Lubrol PX - 582 64,000 0.006 1.0 x 10-4 Triton X-100 - 650 90,000 0.021 3.0 x 10-4 Nonident P-40 - 603 90,000 0.017 3.0 x 10-4 Tween 80
Yeast Nuclear Extract (Small Scale)
Hahn Lab (adapted from J.Leatherwood,Ptashne lab) last modified Mon,Aug 27,2001 Cell Growth 3 liters of cells are grown in YPD (3% glucose)to A600 of 3-5.Antifoam A (two drops from a P200 pipetman)is added to media before autoclaving. For wild
Yeast Nuclear Extract (Small Scale)
Yeast Nuclear Extract (Small Scale) Hahn Lab (adapted from J.Leatherwood,Ptashne lab) last modified Mon,Aug 27,2001 Cell Growth 3 liters of cells are grown in YPD (3% glucose)to A600 of 3-5.Antifoam A (two drops from a P200 pipetman)is added
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