CCK-B Receptor Antagonist 2,15

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CCK-B Receptor Antagonist 2

CAS No. : 155412-88-7

MCE 国际站：CCK-B Receptor Antagonist 2

产品活性：CCK-B Receptor Antagonist 2，化合物 15b，是有效的口服活性 Gastrin/CCK-B 拮抗剂，IC₅₀ 值为 0.43 nM。 CCK-B Receptor Antagonist 2 还抑制 Gastrin/CCK-A 活性，IC₅₀ 为 1.82 μM。

研究领域：GPCR/G Protein  |  Neuronal Signaling

作用靶点：Cholecystokinin Receptor

In Vivo: CCK-B Receptor Antagonist 2 (0.1 μmol/kg; intravenous injection) has an inhibition effect on pentagastrin-induced gastric acid secretion in anethsetized rats with an ED₅₀ of 8.3 nmol/kg.

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