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- 技术资料
- 保存条件：
4°C, sealed storage, away from moisture
- 英文名：
SCH 530348 sulfate
- 库存：
货期：1-2天
- 供应商：
MedChemExpress LLC
- CAS号：
705260-08-8
- 规格：
1 mg/5 mg/10 mg/50 mg
| 规格： | 1 mg | 产品价格： | ￥342.0 |
|---|---|---|---|
| 规格： | 5 mg | 产品价格： | ￥900.0 |
| 规格： | 10 mg | 产品价格： | ￥1500.0 |
| 规格： | 50 mg | 产品价格： | ￥4500.0 |
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Vorapaxar sulfate
CAS No. : 705260-08-8
MCE 国际站：Vorapaxar sulfate
产品活性：Vorapaxar sulfate (SCH 530348 sulfate)，抗血小板活性分子，是一种选择性、口服活性和竞争性的凝血酶受体蛋白酶激活受体 (PAR-1) 拮抗剂，Ki 值为 8.1 nM。Vorapaxar sulfate剂量依赖性抑制凝血酶受体激活肽 (TRAP) 诱导的血小板聚集。
研究领域：GPCR/G Protein
作用靶点：Protease Activated Receptor (PAR)
In Vitro: Vorapaxar sulfate (SCH 530348 sulfate) shows potent inhibition of thrombin-induced platelet aggregation with an IC50 of 47 nM and haTRAP-induced platelet aggregation with an IC50 of 25 nM. Vorapaxar sulfate (SCH 530348 sulfate) inhibits thrombininduced calcium transient in human coronary artery smooth muscle cells (HCASMC) with a Ki of 1.1 nM. It also inhibits thrombin-stimulated thymidine incorporation in HCASMC with a Ki of 13 nM.
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