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- 保存条件:
Powder: -20°C, 3 years; 4°C, 2 years.In solvent: -80°C, 6 months; -20°C, 1 month.
- 库存:
货期:1-2天
- 供应商:
MedChemExpress LLC
- 规格:
10 mM * 1 mL/5 mg/10 mg/50 mg/100 mg
| 规格: | 10 mM * 1 mL | 产品价格: | ¥550.0 |
|---|---|---|---|
| 规格: | 5 mg | 产品价格: | ¥312.0 |
| 规格: | 10 mg | 产品价格: | ¥500.0 |
| 规格: | 50 mg | 产品价格: | ¥1200.0 |
| 规格: | 100 mg | 产品价格: | ¥2000.0 |
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Megestrol
CAS No. : 3562-63-8
MCE 国际站:Megestrol
产品活性:Megestrol 是一种合成的孕激素,用于患有获得性免疫缺陷综合症诊断的患者的厌食症,恶疾或无法解释的重大体重减轻。
研究领域:Metabolic Enzyme/Protease
作用靶点:Drug Metabolite
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文献和实验-羟孕酮类从黄体酮衍生而得。如醋酸甲羟孕酮(醋酸甲孕酮,安宫黄体酮,medroxyprogesterone acetate)、甲地孕酮(megestrol)、氯地孕酮(chlormadinone)和羟孕酮已酸酯(17α-hydroxyprogesterone caproate)。 2.19-去甲睾丸酮类从妊娠素衍生而得。如炔诺酮(norethisterone,norethindrone, norlutin)、双醋炔诺醇(etynodiol diacetate)、炔诺孕酮(18甲基炔诺酮
】孕激素类按化学结构可分为两大类: 1.17α-羟孕酮类从黄体酮衍生而得。如醋酸甲羟孕酮(醋酸甲孕酮,安宫黄体酮,medroxyprogesterone acetate)、甲地孕酮(megestrol)、氯地孕酮(chlormadinone)和羟孕酮已酸酯(17α-hydroxyprogesterone caproate)。 2.19-去甲睾丸酮类从妊娠素衍生而得。如炔诺酮(norethisterone,norethindrone, norlutin)、双醋
。 甲地孕酮醋酸酯(megestrol acetate) 口服,2~4mg/次,1次/日。 炔诺酮(norethisterone) 口服,1.25~5mg/次,1次/日。 丙酸睾酮(testosterone propionate) 肌内注射,10~50mg/日,1~3次/周。 甲睾酮(methyltestosterone) 舌下给药或口服,5~10mg/次,1~2次/日。 苯乙酸睾酮(testosterone phenylacetate)肌内注射。效力较丙酸
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