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IOX4
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Powder: -20°C, 3 years; 4°C, 2 years. In solvent: -80°C, 6 months; -20°C, 1 month.
货期:1-2天
MedChemExpress LLC
10 mM * 1 mL/5 mg/10 mg/50 mg/100 mg
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CAS No. : 1154097-71-8
MCE 国际站:IOX4
产品活性:IOX4 是一种选择性 PHD2 抑制剂,IC50 值为 1.6 nM,在细胞和野生型小鼠中诱导 HIFα 表达,可通透血脑屏障。IOX4 与 PHD2 活性位点的 2-氧代戊二酸 (2OG) 竞争并置换。
研究领域:Metabolic Enzyme/Protease
作用靶点:HIF/HIF Prolyl-Hydroxylase
In Vitro: IOX4 (1-100 μM;5 小时) 确定 HIF1α 诱导的 MCF-7、Hep3B 和 U2OS 中 EC50 分别为 114 μM、86 μM 和 49.5 μM。
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