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- 详细信息
- 文献和实验
- 技术资料
- 保存条件:
Powder: -20°C, 3 years.In solvent: -80°C, 6 months; -20°C, 1 month.
- 库存:
货期:1-2天
- 供应商:
MedChemExpress LLC
- CAS号:
361203-06-7
- 规格:
10 mM * 1 mL/1 mg/5 mg/10 mg
| 规格: | 10 mM * 1 mL | 产品价格: | ¥4059.0 |
|---|---|---|---|
| 规格: | 1 mg | 产品价格: | ¥1470.0 |
| 规格: | 5 mg | 产品价格: | ¥3690.0 |
| 规格: | 10 mg | 产品价格: | ¥5900.0 |
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GW7604
CAS No. : 361203-06-7
MCE 国际站:GW7604
产品活性:GW7604 是一种抗雌激素药。GW7604 是 GW5638 的代谢物。GW5638 是一种高亲和力的雌激素受体 (ER) 拮抗剂。
研究领域:Vitamin D Related/Nuclear Receptor
作用靶点:Estrogen Receptor/ERR
In Vitro: GW7604 is the presumed metabolite of GW5638 in breast (MCF-7) and endometrial (ECC-1) cell lines. GW7604 (0.1 nM-1 μM; 24 hours) inhibits both Estradiol (1 nM) and 4-hydroxytamoxifen (4-OHT; 10 and 100 nM) induction of TGF-alpha in a concentration related manner (1-1000 nM) in MDA-MB-231 cells.
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