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货期:询盘
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MedChemExpress LLC
- CAS号:
2158297-63-1
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询盘
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KRAS G12C inhibitor 5
CAS No. : 2158297-63-1
MCE 国际站:KRAS G12C inhibitor 5
产品活性:KRAS G12C inhibitor 5 是一种 KRas G12C 抑制剂,详细信息请参考专利文献 WO2017201161A1 中的化合物 147。
研究领域:GPCR/G Protein
作用靶点:Ras
In Vitro: Kirsten Rat Sarcoma 2 Viral Oncogene Homolog (KRas) is a small GTPase and a member of the Ras family of oncogenes. KRas serves a molecular switch cycling between inactive (GDP -bound) and active (GTP -bound) states to transduce upstream cellular signals received from multiple tyrosine kinases to downstream effectors to regulate a wide variety of processes, including cellular proliferation.
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