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479080-38-1
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OT antagonist 1
CAS No. : 479080-38-1
MCE 国际站：OT antagonist 1
产品活性：OT antagonist 1 (Compound 4) 是一种有效的选择性催产素 (Oxytocin) 拮抗剂，Ki 为 50 nM。
研究领域：GPCR/G Protein
作用靶点：Oxytocin Receptor
In Vitro: Oxytocin (OT) is a nonapeptide hormone that acts on the OT receptor, a seven-transmembrane (7TM) (Gq-coupled) receptor. The OT receptor has no subtypes but is related to the vasopressin receptors V1A, V1B and V2. OT antagonists have therapeutic potential in a number of areas including pre-term labour: Benign Prostatic Hyperplasia and sexual dysfunction. As a result there is significant interest in the identification of potent, selective, orally bioavailable OT antagonists.
相关产品：Oxytocin acetate | Atosiban acetate | L-368,899 hydrochloride | LIT-001 | Carbetocin | L-371,257 | (Thr4,Gly7)-Oxytocin | Retosiban | Cligosiban | OT-R antagonist 2 | SHR1653 | TC OT 39 | [Asp5]-Oxytocin | (d(CH2)51,Tyr(Me)2,Orn8)-Oxytocin | (d(CH2)51,Tyr(Me)2,Thr4,Orn8,des-Gly-NH29)-Vasotocin | (d(CH2)51,Tyr(Me)2,Thr4,Orn8,Tyr-NH29)-Vasotocin | (Val3,Pro8)-Oxytocin | Barusiban | Cargutocin | Demoxytocin | L-366682 | L-372662 | PF-06478939
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文献和实验for the treatment of SCLC (1 ,2) . Although antagonist G blocks SCLC cell growth (IC50 = 24.5 � 1.5 and 38.5 � 1.5 μM for the H69 and H510 cell lines, respectively), its exact mechanism of action is unclear. Factors affecting the balance between SCLC cell
Characterization of Histaminergic Receptors
‐methyl histamine >100,000 >100,000 38 – RBI H 1 Antagonists Chlorpheniramine 7.6 6100 1500 – RBI Diphenhydramine 17 2500 >10,000 >10,000
like PKB. Proapoptotic proteins which can be phosphorylated and inhibited by PKB include BAD (BCL2 Antagonist of Cell Death), human Caspase9, and the forkhead family of transcription factors. PKB can also cause stimulation of NF-KappaB (Nuclear Factor-Kappa
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