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JTE-952
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4°C, sealed storage, away from moisture and light
货期:1-2天
MedChemExpress LLC
10 mM * 1 mL/1 mg/5 mg/10 mg
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CAS No. : 1255303-54-8
MCE 国际站:JTE-952
产品活性:JTE-952 是 集落刺激因子-1 受体 (CSF-1R/cFMS) 有效的、具有口服活性的、 II 型 选择性抑制剂,其对 CSF1R 和 TrkA 的IC50 值分别为 13 nM 和 261 nM。可用于关节炎的相关研究。
研究领域:Protein Tyrosine Kinase/RTK
作用靶点:c-Fms
In Vivo: JTE-952 (3 mg/kg, p.o. once-daily) treatment reduces the overall progression of the clinical score, including inflammation and bone erosion in mouse model of collagen-induced arthritis (CIA model).
相关产品:Bioactive Compound Library Plus | Immunology/Inflammation Compound Library | Kinase Inhibitor Library | Protein Tyrosine Kinase Compound Library | Coagulation and Anti-coagulation Compound Library | Pain-Related Compound Library | Membrane Protein-targeted Compound Library | Highly Selective Inhibitors Library | Cytokine Inhibitors Library | Pexidartinib | PLX5622 | Sotuletinib | Linifanib | Dovitinib | GW2580 | PLX5622 in AIN-76A Diet (1200 ppm) | Pazopanib Hydrochloride | Edicotinib | Vimseltinib | Chiauranib | PLX647 | Elzovantinib | Seralutinib | Emactuzumab | PRN1371 | c-Fms-IN-1 | Ki20227 | AZD7507 | BPR1R024 | CSF1R-IN-1 | OSI-930 | Mavrilimumab | cFMS Receptor Inhibitor II | CSF1R-IN-3 | c-Fms-IN-10 | c-Fms-IN-13
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