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- 详细信息
- 文献和实验
- 技术资料
- 库存:
361
- 英文名:
Neratinib
- CAS号:
698387-09-6
- 保质期:
2年
- 供应商:
北京百奥莱博科技有限公司
- 保存条件:
-20℃,有效期2年,溶入溶剂后-20℃
- 规格:
1mL(10mM)|5mg|10mg|50mg|100mg|200mg
特别提示:包括tyrosine kinase抑制剂(Neratinib)在内,本公司的所有产品仅可用于科研实验,严禁用于临床医疗及其他非科研用途!
产品名称:tyrosine kinase抑制剂(Neratinib)
英文名称:Neratinib
产品货号:M00234
产品规格:1mL(10mM)|5mg|10mg|50mg|100mg|200mg
Neratinib是一种可,不可逆的tyrosine kinase抑制剂,能够抑制HER2和EGFR的活性,IC50值分别为59nM和92nM。
注:本品仅可用于科研实验,严禁用于临床医疗及其他用途!
CAS号:698387-09-6
别名:HKI-272
纯度:99.54%
分子式:C₃₀H₂₉ClN₆O₃
分子量:557.04
结构式:
储存条件:-20℃,有效期2年,溶入溶剂后-20℃请尽量在一个月内使用。
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文献和实验phosphorylation, and downmodulate cellular protein tyrosine kinase activities (1 –6 ). These LMP2A functional studies have involved in vitro assays to determine the phosphorylation patterns of both LMP2A and cellular signal transducers before and after BCR
Analysis of Janus Tyrosine Kinase Phosphorylation and Activation
-phosphotyrosine-directed Western blot analysis of Jak-specific immunoprecipitates. Additionally, receptor pull-down and in vitro kinase assays can also be utilized to measure cellular Jak catalytic activity. In addition to tyrosine phosphorylation, recent evidence
Tyrosine Kinase Inhibitors Against EGF Receptor-Positive Malignancies
epidermal growth factor receptor (EGFR) (1 –6 ), Janus kinases (JAKs) (7 –13 ), Bruton’s tyrosine kinase (BTK) (14 –16 ), platelet-derived growth factor (PDGF) (17 ), protein kinase C (PKC) (18 –24 ), Lck (25 , 26 ), Trk (27 –30
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