一种脂联素受体激动剂,能够与 AdipoR1 和 AdipoR2 结合。AdipoRon is an adiponectin receptor (AdipoR) agonist and binds to AdipoR1 and AdipoR2 at low μm concentration. AdipoRon activates AMPK (5'-adenosine monophosphate-activated protein kinase ) in cultured mammalian cells and activates PGC-1 (peroxisome proliferator-activated receptor γ coactivator 1-α) which boosts mitochondrial proliferation and energy metabolism.