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- 2025年12月04日
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- 详细信息
- 技术资料
- 保存条件：
Powder: -20°C, 3 years; 4°C, 2 years.In solvent: -80°C, 6 months; -20°C, 1 month.
- 库存：
货期：1-2天
- 供应商：
MedChemExpress LLC
- CAS号：
1186430-60-3
- 规格：
10 mM * 1 mL/5 mg/10 mg/25 mg/50 mg/100 mg
| 规格： | 10 mM * 1 mL | 产品价格： | ￥753.0 |
|---|---|---|---|
| 规格： | 5 mg | 产品价格： | ￥684.0 |
| 规格： | 10 mg | 产品价格： | ￥1185.0 |
| 规格： | 25 mg | 产品价格： | ￥2038.0 |
| 规格： | 50 mg | 产品价格： | ￥3260.0 |
| 规格： | 100 mg | 产品价格： | ￥5200.0 |
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Antihistamine-1
CAS No. : 1186430-60-3
MCE 国际站：Antihistamine-1
产品活性：Antihistamine-1 是能够渗透血脑屏障的 H1-抗组胺药 (Ki=6.9 nM), 它也是 CYP2D6 和 hERG 通道的抑制剂，其 IC50 值分别为 5.4 和 0.8 μM。
研究领域：GPCR/G Protein | Neuronal Signaling | Immunology/Inflammation | Metabolic Enzyme/Protease | Membrane Transporter/Ion Channel
作用靶点：Histamine Receptor | Cytochrome P450 | Potassium Channel
In Vitro: Antihistamine-1 (Compound 2) is a H1-antihistamine (Ki=6.9 nM) with acceptable blood-brain barrier penetration and also an inhibitor of CYP2D6 and hERG channel with IC50s of 5.4 and 0.8 μM, respectively.
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