Cabergoline

概述

• 产品名称
  Cabergoline
• 描述
  D₂-like receptor agonist
• 生物学描述
  D₂-like receptor agonist (K_i values are 0.7 (D₂), 1.5 (D₃), 9.0 (D₄) and 165 nM (D₅)). Highly potent at some 5-HT receptors (K_i values are 20 (5-HT_1A), 8.7 (5-HT_1D), 6.2 (5-HT_2A) and 1.2 nM (5-HT_2B)). Shows antitumour effects and has antidepressant and anxiolytic properties.
• 纯度
  > 99%

性能

• 化学名称
  N-[3-(Dimethylamino)propyl]-N-[(ethylamino)carbonyl]-6-(2-propenyl)ergoline-8β-carboxamide
• 分子量
  451.60
• 化学结构
  
• 分子式
  C₂₆H₃₇N₅O₂
• CAS编号
  81409-90-7
• 存放说明
  Store at +4°C. The product can be stored for up to 12 months.
• 溶解度概述
  Soluble in ethanol to 100 mM and in DMSO to 100 mM
• 处理

  Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.

  Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.

• 来源

  Synthetic