HY-70005 |
CPA inhibitor |
CPA inhibitor是羧肽酶A(CPA)抑制剂。 |
223532-02-3 |
carboxypeptidase inhibitor;Benzenepropanoic acid, .alpha.-[[hydroxy(2-phenylacetyl)amino]methyl]- |
HY-70006 |
TOK-001 |
TOK-001 (VN/124-1; Galeterone)是多功能抗雄激素和CYP17抑制剂,IC50为47 nM。 |
851983-85-2 |
VN/124-1; Galeterone; VN 124;TOK001;TOK 001 |
HY-70083 |
SPK-601 |
SPK-601(LMV-601)是卵磷脂特异磷脂酶C(PC-PLC)抑制剂,可用作抗菌剂。 |
1096687-52-3 |
LMV-601;SPK601;SPK 601 |
HY-70027 |
p53 and MDM2 proteins-interaction-inhibitor (chiral) |
手性p53 and MDM2 proteins-interaction-inhibitor是p53和MDM2相互作用的抑制剂。 |
939981-37-0 |
p53 inhibitor (chiral); Ethanone, 2-[4-[[(4S,5R)-4,5-bis(4-chlorophenyl)-2-[4-(1,1-dimethylethyl)-2-ethoxyphenyl]-4,5-dihydro-4,5-dimethyl-1H-imidazol-1-yl]carbonyl]-1-piperazinyl]-1-(4-morpholinyl)- |
HY-70028 |
p53 and MDM2 proteins-interaction-inhibitor (racemic) |
外消旋p53 and MDM2 proteins-interaction-inhibitor是p53与MDM2相互作用抑制剂。 |
939983-14-9 |
p53 inhibitor (racemic); Ethanone, 2-[4-[[(4R,5S)-4,5-bis(4-chlorophenyl)-2-[4-(1,1-dimethylethyl)-2-ethoxyphenyl]-4,5-dihydro-4,5-dimethyl-1H-imidazol-1-yl]carbonyl]-1-piperazinyl]-1-(4-morpholinyl)-, rel- |
HY-10959 |
RG7112 |
RG7112是第一个进入临床的MDM2抑制剂,能占据MDM2上与p53结合的活性口袋。 |
939981-39-2 |
RG-7112;RG 7112 |
HY-10043 |
gamma-secretase modulator 1 |
γ-secretase inhibitior-1是γ-secretase调节剂,可作用于阿尔茨海默病。 |
1172637-87-4 |
2-Benzothiazolamine, 4,5,6,7-tetrahydro-N-[3-methoxy-4-(4-methyl-1H-imidazol-1-yl)phenyl]-4-phenyl- |
HY-50865 |
PDE-9 inhibitor |
PDE-9抑制剂可作用于神经退行性疾病。 |
1082743-70-1 |
PDE-9 ; PDE 9 ;4H-Pyrazolo[3,4-d]pyrimidin-4-one, 1,5-dihydro-6-[(3S,4S)-4-methyl-1-(phenylmethyl)-3-pyrrolidinyl]-1-(tetrahydro-2H-pyran-4-yl)- |
HY-50859 |
Ruxolitinib (sulfate) |
Ruxolitinib(INCB018424)硫酸盐是第一个进入临床的高活性JAK1和2选择性抑制剂,IC50分别为3.3 nM和2.8 nM,比对JAK3的抑制性高130倍以上。 |
1092939-16-6 |
INCB018424 sulfate;INCB 018424 sulfate;INCB-018424 sulfate;Ruxolitinib |
HY-50858 |
Ruxolitinib (phosphate) |
Ruxolitinib(INCB018424)磷酸盐是第一个进入临床的高活性JAK1和2选择性抑制剂,IC50分别为3.3 nM和2.8 nM,比对JAK3的抑制性高130倍以上。 |
1092939-17-7 |
INCB018424 phosphate;INCB 018424 phosphate;INCB-018424 phosphate;Ruxolitinib |