相关产品推荐更多 >
万千商家帮你免费找货
0 人在求购买到急需产品
- 详细信息
- 技术资料
- 保存条件:
Powder: -20°C, 3 years; 4°C, 2 years.In solvent: -80°C, 6 months; -20°C, 1 month.
- 英文名:
MK-3102
- 库存:
货期:1-2天
- 供应商:
MedChemExpress LLC
- 规格:
10 mM * 1 mL/1 mg/2 mg/5 mg/10 mg/25 mg/50 mg
| 规格: | 10 mM * 1 mL | 产品价格: | ¥1016.0 |
|---|---|---|---|
| 规格: | 1 mg | 产品价格: | ¥486.0 |
| 规格: | 2 mg | 产品价格: | ¥700.0 |
| 规格: | 5 mg | 产品价格: | ¥1159.0 |
| 规格: | 10 mg | 产品价格: | ¥1900.0 |
| 规格: | 25 mg | 产品价格: | ¥3650.0 |
| 规格: | 50 mg | 产品价格: | ¥5413.0 |
MCE 的所有产品仅用作科学研究或药证申报,我们不为任何个人用途提供产品和服务。
Omarigliptin
CAS No. : 1226781-44-7
MCE 国际站:Omarigliptin
产品活性:Omarigliptin (MK-3102) 是一种有效的、选择性的、具有口服活性的并能穿过血脑屏障的二肽基肽酶 4 dipeptidyl peptidase 4 (DPP-4) 抑制剂。Omarigliptin 显示出抗帕金森病活性。Omarigliptin 具有改善糖尿病相关认知功能障碍的神经保护作用。
研究领域:Metabolic Enzyme/Protease
作用靶点:Dipeptidyl Peptidase
In Vivo: Omarigliptin (5 mg/kg; p.o.) enhances the intestinal glucagon like peptide-1 and crosses BBB in rats.
Omarigliptin (2.5, 5 mg/kg; p.o.; once a week for 8 weeks) shows anti-diabetic activity in STZ-induced diabetic mice.
Omarigliptin (5 mg/kg; p.o.; daily for 28 days) shows anti-parkinsonian activity in rats.
相关产品:Covalent Screening Library Plus | Drug Repurposing Compound Library Plus | FDA-Approved Drug Library Plus | FDA-Approved Drug Library Mini | Bioactive Compound Library Plus | Metabolism/Protease Compound Library | FDA-Approved Drug Library | CNS-Penetrant Compound Library | Drug Repurposing Compound Library | Covalent Screening Library | Anti-diabetic Compound Library | Ferroptosis Compound Library | Anti-COVID-19 Compound Library | Orally Active Compound Library | FDA Approved & Pharmacopeial Drug Library | Neuroprotective Compound Library | Anti-Parkinson's Disease Compound Library | Neurodegenerative Disease-related Compound Library | Heterocyclic Compound Library | Highly Selective Inhibitors Library | Puromycin aminonucleoside | Sitagliptin | Talabostat mesylate | Linagliptin | Brensocatib | Saxagliptin | 1G244 | Vildagliptin | Diprotin A | Teneligliptin | Nateglinide | Alogliptin | Trelagliptin | Anagliptin | Gemigliptin tartrate | DPP-IV-IN-2 | Retagliptin phosphate | UAMC00039 dihydrochloride | DPP-IV-IN-1 | Azaleatin | DBPR108 | Dutogliptin | Evogliptin tartrate | NDMC101
热门产品线:重组蛋白 | 化合物库 | 天然产物 | 荧光染料 | PROTAC | 同位素标记物
Trending products:Recombinant Proteins | Bioactive Screening Libraries | Natural Products | Dye Reagents | PROTAC | Isotope-Labeled Compounds
风险提示:丁香通仅作为第三方平台,为商家信息发布提供平台空间。用户咨询产品时请注意保护个人信息及财产安全,合理判断,谨慎选购商品,商家和用户对交易行为负责。对于医疗器械类产品,请先查证核实企业经营资质和医疗器械产品注册证情况。
技术资料暂无技术资料 索取技术资料


















