LH846,639052-78-1

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LH846

CAS No. : 639052-78-1

MCE 国际站：LH846

产品活性：LH846 是一种选择性的 CKIδ 抑制剂，IC₅₀ 值为 290 nM；对 CKIα 和 CKIε 的抑制作用相对较弱，IC₅₀ 值分别为 2.5 μM 和 1.3 μM。

研究领域：Cell Cycle/DNA Damage  |  Stem Cell/Wnt

作用靶点：Casein Kinase

In Vitro: LH846 is a potent inhibitor of CKIδ, with an IC₅₀ of 290 nM, less potently inhibits CKIα and CKIε, with IC₅₀s of 2.5 μM and 1.3 μM, respectively, and has no effect on CK2. LH846 (3 or 10 μM) inhibits CKIδ-dependent phosphorylation of PER1 in HEK293T cells.

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