Leuprolide Acetate

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Leuprolide Acetate

CAS No. : 74381-53-6

MCE 国际站：Leuprolide Acetate

产品活性：Leuprolide Acetate (Leuprorelin acetate) 是一种促性腺激素释放激素 (GnRH) 类似物，能作为 GnRH 受体 (GnRH receptor) 激动剂。Leuprolide Acetate 可用于前列腺癌、子宫内膜异位症、子宫肌瘤、中枢性早熟、多发性硬化症的研究。Leuprolide Acetate 能改善大鼠模型中的实验性自身免疫性脑脊髓炎 (EAE)。

研究领域：GPCR/G Protein

作用靶点：GNRH Receptor

In Vitro: Leuprolide Acetate (0.01 nM-μM; 6-30 days) induces a significant increase in the GnRH receptor levels.

In Vivo: Leuprolide Acetate (1.2 μg/kg; i.m.; 5 application times) decreases the severity of clinical signs of locomotion, induces a significantly greater body weight gain, increases the MBP and NFs expression, axonal area and cell infiltration in (EAE) rats.

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