8-Cyclopentyl-1,3-dipropylxant

1) Cat. No.: TRC-C988500; 2) Chemical Name: 8-Cyclopentyl-1,3-dipropylxanthine; 3) CAS No.: 102146-07-6; 4) Mol. Formula: C16H24N4O2; 5) Mol. Weight: 304.39; 6) Packing Size: 100mg / 1g; 7) Appearence: White Solid; 8) Application Notes: DPCPX is a potent and very selective A1-adenosine receptor antagonist, with a Ki of 0.46 nM for A1 receptors in rat whole-brain membranes. Its 740-fold A1-selectivity is the highest reported for an adenosine antagonist.; 9) Synonym: 8-Cyclopentyl-3,9-dihydro-1,3-dipropyl-1H-purine-2,6-dione; DPCPX, PD 116,948; 10) Solubility: DMSO (3.6 mg/ml), Ethanol (4 mg/ml), 0.1N Sodium Hydroxide (2 mg/ml); 11) Storage condition: -20˚C Freezer; 12) References: Gessi, S., et al.: Mol. Pharmacol., 67, 2137 (2005), Minor, T.R., et al.: Behav. Neurosci., 122, 1236 (2008), Gracia, E., et al.: J. Neurochem., 107, 161 (2008), Gessi, S., et al.: Biochem. Pharmacol., 75, 562 (2008),