AR-C155858

1) Cat. No.: TRC-A187720; 2) Chemical Name: AR-C155858 ; 3) CAS No.: ; 4) Mol. Formula: 461.53; 5) Mol. Weight: 212755; 6) Packing Size: 5mg / 50mg; 7) Appearence: ; 8) Application Notes: AR-C155858 is a potent inhibitor of monocarboxylate transporters MCT1 and MCT2 that binds to an intracellular site involving transmembrane helices 7-10.; 9) Synonym: (S)-6-[(3,5-Dimethyl-1H-pyrazol-4-yl)methyl]-5-[(4-hydroxyisoxazolidin-2-yl)carbonyl]-1-isobutyl-3-methylthieno[2,3-d]pyrimidine-2,4(1H,3H)-dione; 2-[[6-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,2,3,4-tetrahydro-3-methyl-1-(2-methylpropyl)-2,4-dioxothieno[2,3-d]pyrimidin-5-yl]carbonyl]-4-isoxazolidinol; (S)-6-[(3,5-Dimethyl-1H-pyrazol-4-yl)methyl]-5-[(4-hydroxyisoxazolidin-2-yl)carbonyl]-1-isobutyl-3-methylthieno[2,3-d]pyrimidine-2,4(1H,3H)-dione; AR-C 155858 ; 10) Solubility: ; 11) Storage condition: ; 12) References: Ovens, M.J., et al.: Biochem. J., 425, 523 (2010);