- ￥1215 - 2813
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- D57901
- 2025年10月17日
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1mg/5mg
| 规格： | 1mg | 产品价格： | ￥1215.0 |
|---|---|---|---|
| 规格： | 5mg | 产品价格： | ￥2813.0 |
| 产品编号 | D57901 |
| 英文名称 | (E)-GABAB receptor antagonist 1 |
| 中文名称 | (E)-GABAB受体拮抗剂-1 |
| 理论分子量 | 304.38 |
| 保存条件 | Powder: -20℃ for 3 years | In solvent: -80℃ for 1 year |
| 注意事项 | This product as supplied is intended for research use only, not for use in human, therapeutic or diagnostic applications. |
| 背景资料 | (E)-GABAB receptor antagonist 1 is a trans-GABAB receptor antagonist 1. (E)-GABAB receptor antagonist 1 decreases GABA-induced IP3 (inositol trisphosphate) production with IC50 of 37.9 μM. GABAB receptor antagonist 1 is a selective and negative allosteric modulator of GABAB (γ-Aminobutyric acid) receptors. |
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文献和实验[3H](+)MK801 Radioligand Binding Assay at the N‐Methyl‐D‐Aspartate Receptor
. Bonhaus, D.W. and McNamara, J.O. 1998. N‐methyl‐D‐aspartate receptor regulation of uncompetitive antagonist binding in rat brain membranes: Kinetic analysis. Mol. Pharmacol. 34:250‐255
Overview of Receptor Allosterism
Spalding, T.A., Trotter, C., Skjaerbaek, N., Messier, T.L., Currier, E.A., Burstein, E.S., Li, D., Hacksell, U., and Brann, M.R. 2002. Discovery of an ectopic activation site on the M(1) muscarinic receptor. Mol. Pharmacol. 61:1297‐1302
[D-Arg6 , D-Trp7,9 , Nme Phe8 ]-substance P (6-11) (antagonist G) is a novel class of anti-cancer agent that inhibits small cell lung cancer (SCLC) cell growth in vitro and in vivo and is entering Phase II clinical investigation
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