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- 保存条件:
-20°C
- 保质期:
咨询
- 英文名:
Deferasirox
- 库存:
1000+
- 供应商:
上海维亦特生物
- CAS号:
201530-41-8
纯度:>98% by HPLC;NMR (Conforms)
分子式:C21H15N3O4
分子量:373.36
溶剂:DMSO (10 mg/ml)
性状:Off-white to white solid
存储:-20°C
Activity (short version):Iron chelator
Function / Pharmacology:Clinically useful iron chelator used in long term care of ß-thalassemia and other heavily transfused hematological patients.1,2 It has been shown to potent inhibitor of JumonjiC Domain-Containing Histone Demethylases (IC50’s = KDM4A(JMJD2A) 4.76 µM, KDM5A(JARID1A) 5.00 µM, KDM6B(JMJD3) 3.95 µM).3 Deferasirox has also been investigated as a potential anticancer agent.4-6
分子式:C21H15N3O4
分子量:373.36
溶剂:DMSO (10 mg/ml)
性状:Off-white to white solid
存储:-20°C
Activity (short version):Iron chelator
Function / Pharmacology:Clinically useful iron chelator used in long term care of ß-thalassemia and other heavily transfused hematological patients.1,2 It has been shown to potent inhibitor of JumonjiC Domain-Containing Histone Demethylases (IC50’s = KDM4A(JMJD2A) 4.76 µM, KDM5A(JARID1A) 5.00 µM, KDM6B(JMJD3) 3.95 µM).3 Deferasirox has also been investigated as a potential anticancer agent.4-6
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文献和实验该产品被引用文献
201530-41-8
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Deferasirox
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