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- 详细信息
- 文献和实验
- 技术资料
- 保存条件:
-20°C
- 保质期:
咨询
- 英文名:
Go-6983
- 库存:
1000+
- 供应商:
上海维亦特生物
- CAS号:
133053-19-7
纯度:98% by HPLC,;NMR (Conforms)
分子式:C26H26N4O3
分子量:442.51
溶剂:DMSO (20 mg/ml)
性状:Red-orange solid
存储:-20°C
Activity (short version):PKC inhibitor
Function / Pharmacology:A potent and pan-specific, ATP-competitive protein kinase C inhibitor. PKC isotype IC50s= 7, 7, 6, 10 and 60 nM for PKC α, β, γ, δ, ζ respectively.1 Suppresses stress induced HSP27 disassociation.2 Maintains rat embryonic stem cell pluripotency.3 Attenuates myocardial ischemia/reperfusion injury.4
分子式:C26H26N4O3
分子量:442.51
溶剂:DMSO (20 mg/ml)
性状:Red-orange solid
存储:-20°C
Activity (short version):PKC inhibitor
Function / Pharmacology:A potent and pan-specific, ATP-competitive protein kinase C inhibitor. PKC isotype IC50s= 7, 7, 6, 10 and 60 nM for PKC α, β, γ, δ, ζ respectively.1 Suppresses stress induced HSP27 disassociation.2 Maintains rat embryonic stem cell pluripotency.3 Attenuates myocardial ischemia/reperfusion injury.4
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文献和实验该产品被引用文献
133053-19-7
相关实验
Spatiotemporal Dynamics of Kinase Signaling Visualized by Targeted Reporters
Activator of kinase signaling path: e.g., histamine or phorbol dibutyrate (PdBu) Kinase inhibitor or inhibitor of kinase signaling pathway, as control: e.g., Gö 6983
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文献支持
Go-6983
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