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- 保存条件:
-20°C
- 保质期:
咨询
- 英文名:
Phosphoramidon
- 库存:
1000+
- 供应商:
上海维亦特生物
- CAS号:
119942-99-3
纯度:97% by TLC;NMR (Conforms)
分子式:C23H32N3O10P·2Na
分子量:587.47
溶剂:DMSO (>25 mg/ml) Water (>25 mg/ml)
性状:White solid
存储:-20°C
Activity (short version):Neutral endopeptidase inhibitor
Function / Pharmacology:Inhibits neutral endopeptidase 24.11 (NEP; Neprilysin; EC 3.4.24.11), Ki=2 nM.1 Also inhibits neprilysin 2 (Ki~2 nM).2 Also inhibits endothelin-converting enzyme (IC50 = 0.68 μM).3 Induces a dramatic increase in amyloid-beta levels in rodents.4
分子式:C23H32N3O10P·2Na
分子量:587.47
溶剂:DMSO (>25 mg/ml) Water (>25 mg/ml)
性状:White solid
存储:-20°C
Activity (short version):Neutral endopeptidase inhibitor
Function / Pharmacology:Inhibits neutral endopeptidase 24.11 (NEP; Neprilysin; EC 3.4.24.11), Ki=2 nM.1 Also inhibits neprilysin 2 (Ki~2 nM).2 Also inhibits endothelin-converting enzyme (IC50 = 0.68 μM).3 Induces a dramatic increase in amyloid-beta levels in rodents.4
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