Galectin-3-IN-4,2496515-38-7

Galectin-3-IN-4

产品活性：Galectin-3-IN-4 (compound 5) 是一种羧酰胺类似物。Galectin-3-IN-4 是一种有效的、选择性的、口服生物可利用的人和小鼠 Galectin-3 抑制剂，对 hGal-3 和 mGal-3 的 IC50 值分别为 21 和 167 nM。 Galectin-3-IN-4 对于 hGal-1 和 hGal-9 的 IC50 值分别为 1580 和 2750 nM[1]。

产品来源： www.medchemexpress.cn/galectin-3-in-4.html

研究领域：Immunology/Inflammation

作用靶点：Galectin

In Vivo: Galectin-3-IN-4 (compound 5) (2 mg/kg IV, 10 mg/kg PO; once) has a low clearance rate (CL = 12 mL/min/kg) and a high volume of distribution (Vss = 2.1 L/kg), and has a 52 % oral bioavailabilities in mice.

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