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- 详细信息
- 技术资料
- 保存条件:
polypeptide, sealed storage, away from moisture
- 库存:
国内:现货
- 供应商:
MedChemExpress LLC
- 规格:
1 mg
HS014 TFA
产品活性:HS014 TFA 是一种高效、选择性的黑素皮质素-4 (MC4) 受体拮抗剂,对人 MC4、MC1、MC3 和 MC5 受体的 Ki 值分别为 3.16、108、54.4 和 694 nM。HS014 TFA 增加自由喂养大鼠的食物摄取量。
产品来源: www.medchemexpress.cn/hs014-tfa.html
研究领域:GPCR/G Protein | Neuronal Signaling
作用靶点:Melanocortin Receptor
In Vivo: Pretreatment with HS014 TFA blocks the effect of IL-1beta on food intake and respiratory exchange ratio (RER) at later time points (beyond 8 h post injection), as well as the hypoactivity and increases metabolic rate.
相关产品:Bioactive Compound Library Plus | Macrocyclic Compound Library | Peptide Library | Cyclic Peptide Library | α-MSH | Melanotan I | SHU 9119 | Bremelanotide Acetate | BMS-470539 dihydrochloride | Nonapeptide-1 acetate salt | Adrenocorticotropic Hormone (ACTH) (1-39), rat TFA | JNJ-10229570 | THIQ | HS024 TFA | β-Melanocyte Stimulating Hormone (MSH), human TFA | PF-00446687 | ACTH (1-17) (TFA) | Adrenocorticotropic Hormone (ACTH) (1-39), human(TFA) | Dersimelagon | MK-0493 | SNT-207707 | SNT-207858 free base | [D-Trp8]-γ-MSH | ACTH (11-24) | Adrenocorticotropic Hormone (ACTH) (4-10), human | Agouti-related Protein (AGRP) (83-132) Amide (human) (TFA) | Fenoprofen | MSG606 | γ-1-Melanocyte Stimulating Hormone (MSH), amide | ML-00253764 hydrochloride | PF-07258669 | PG-931
产品活性:HS014 TFA 是一种高效、选择性的黑素皮质素-4 (MC4) 受体拮抗剂,对人 MC4、MC1、MC3 和 MC5 受体的 Ki 值分别为 3.16、108、54.4 和 694 nM。HS014 TFA 增加自由喂养大鼠的食物摄取量。
产品来源: www.medchemexpress.cn/hs014-tfa.html
研究领域:GPCR/G Protein | Neuronal Signaling
作用靶点:Melanocortin Receptor
In Vivo: Pretreatment with HS014 TFA blocks the effect of IL-1beta on food intake and respiratory exchange ratio (RER) at later time points (beyond 8 h post injection), as well as the hypoactivity and increases metabolic rate.
相关产品:Bioactive Compound Library Plus | Macrocyclic Compound Library | Peptide Library | Cyclic Peptide Library | α-MSH | Melanotan I | SHU 9119 | Bremelanotide Acetate | BMS-470539 dihydrochloride | Nonapeptide-1 acetate salt | Adrenocorticotropic Hormone (ACTH) (1-39), rat TFA | JNJ-10229570 | THIQ | HS024 TFA | β-Melanocyte Stimulating Hormone (MSH), human TFA | PF-00446687 | ACTH (1-17) (TFA) | Adrenocorticotropic Hormone (ACTH) (1-39), human(TFA) | Dersimelagon | MK-0493 | SNT-207707 | SNT-207858 free base | [D-Trp8]-γ-MSH | ACTH (11-24) | Adrenocorticotropic Hormone (ACTH) (4-10), human | Agouti-related Protein (AGRP) (83-132) Amide (human) (TFA) | Fenoprofen | MSG606 | γ-1-Melanocyte Stimulating Hormone (MSH), amide | ML-00253764 hydrochloride | PF-07258669 | PG-931
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HS014 TFA
¥4500










