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- 详细信息
- 技术资料
- 保存条件:
-20°C, protect from light, stored under nitrogen
- 库存:
货期:1-2天
- 供应商:
MedChemExpress LLC
- CAS号:
3036109-10-8
- 规格:
5 mg/10 mg/25 mg
| 规格: | 5 mg | 产品价格: | ¥1700.0 |
|---|---|---|---|
| 规格: | 10 mg | 产品价格: | ¥2730.0 |
| 规格: | 25 mg | 产品价格: | ¥6000.0 |
SDU-071
产品活性:SDU-071 是有效的,有口服活性的 BRD4-p53 抑制剂。SDU-071 抑制 MDA-MB-231 细胞增殖,其IC50 为 10.5 μM。SDU-071 诱导细胞周期阻滞和凋亡 (apoptosis)。
产品来源: www.medchemexpress.cn/sdu-071.html
研究领域:Epigenetics | Apoptosis
作用靶点:Epigenetic Reader Domain | Apoptosis
In Vitro: SDU-071 (10 μM, 24 h) induces cell-cycle arrest and apoptosis in MDA-MB-231 cells.SDU-071 (10 μM, 72 h) inhibits cell proliferation, migration, and invasion in MDA-MB-231 cells.
In Vivo: SDU-071 (250 mg/kg for i.g; once daily for 21 days) inhibits tumor growth in a MDA-MB-231 orthotopic mouse xenograft mammary tumor model.
相关产品:MG-132 | Doxorubicin hydrochloride | Bafilomycin A1 | Tamoxifen | Y-27632 | LY294002 | Paclitaxel | Z-VAD-FMK | Acetylcysteine | Angiotensin II human | 2-Deoxy-D-glucose | Staurosporine | Actinomycin D | SB-431542 | 5-Fluorouracil | Bortezomib | Deferoxamine mesylate | Oxaliplatin | Trametinib | Sorafenib | Temozolomide | Gemcitabine | Decitabine | Mdivi-1 | Elesclomol | Rotenone | Etoposide | Ruxolitinib | SP600125 | Monomethyl auristatin E
产品活性:SDU-071 是有效的,有口服活性的 BRD4-p53 抑制剂。SDU-071 抑制 MDA-MB-231 细胞增殖,其IC50 为 10.5 μM。SDU-071 诱导细胞周期阻滞和凋亡 (apoptosis)。
产品来源: www.medchemexpress.cn/sdu-071.html
研究领域:Epigenetics | Apoptosis
作用靶点:Epigenetic Reader Domain | Apoptosis
In Vitro: SDU-071 (10 μM, 24 h) induces cell-cycle arrest and apoptosis in MDA-MB-231 cells.SDU-071 (10 μM, 72 h) inhibits cell proliferation, migration, and invasion in MDA-MB-231 cells.
In Vivo: SDU-071 (250 mg/kg for i.g; once daily for 21 days) inhibits tumor growth in a MDA-MB-231 orthotopic mouse xenograft mammary tumor model.
相关产品:MG-132 | Doxorubicin hydrochloride | Bafilomycin A1 | Tamoxifen | Y-27632 | LY294002 | Paclitaxel | Z-VAD-FMK | Acetylcysteine | Angiotensin II human | 2-Deoxy-D-glucose | Staurosporine | Actinomycin D | SB-431542 | 5-Fluorouracil | Bortezomib | Deferoxamine mesylate | Oxaliplatin | Trametinib | Sorafenib | Temozolomide | Gemcitabine | Decitabine | Mdivi-1 | Elesclomol | Rotenone | Etoposide | Ruxolitinib | SP600125 | Monomethyl auristatin E
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SDU-071,3036109-10-8
¥1700 - 6000










