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Please store the product under the recommended conditions in the Certificate of Analysis.
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货期:询盘
- 供应商:
MedChemExpress LLC
- CAS号:
2100855-80-7
- 规格:
询盘
PI3Kα-IN-1
产品活性:PI3Kα-IN-1 是一种 PI3Kα 抑制剂 (IC50 IC 50: 104 nM)。
产品来源: www.medchemexpress.cn/pi3kα-in-1.html
研究领域:PI3K/Akt/mTOR
作用靶点:PI3K
In Vitro: PI3Kα-IN-1 shows good stability in the mouse liver microsome assay (t1/2 values > 60 minutes).PI3Kα-IN-1 (48 h) induces cytotoxicity in MDC7 cells with an IC50 value of around 170 nM.PI3Kα-IN-1 (15-250 nM) inhibits phospho4EBP, phosphor-P70SK6 and phospho-473AKT in MCF7 cells.
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产品活性:PI3Kα-IN-1 是一种 PI3Kα 抑制剂 (IC50 IC 50: 104 nM)。
产品来源: www.medchemexpress.cn/pi3kα-in-1.html
研究领域:PI3K/Akt/mTOR
作用靶点:PI3K
In Vitro: PI3Kα-IN-1 shows good stability in the mouse liver microsome assay (t1/2 values > 60 minutes).PI3Kα-IN-1 (48 h) induces cytotoxicity in MDC7 cells with an IC50 value of around 170 nM.PI3Kα-IN-1 (15-250 nM) inhibits phospho4EBP, phosphor-P70SK6 and phospho-473AKT in MCF7 cells.
相关产品:3-Methyladenine | LY294002 | Quercetin | Alpelisib | 740 Y-P | Wortmannin | AZD-7648 | Buparlisib | Copanlisib | Pictilisib | Dactolisib | Idelalisib | Inavolisib | SAR405 | Duvelisib | α-Linolenic acid | Eganelisib | YM-201636 | Omipalisib | Recilisib | Isorhamnetin | PI-103 | Taselisib | Fimepinostat | Vps34-IN-1 | GSK2636771 | 1-Deoxynojirimycin | hSMG-1 inhibitor 11j | iMDK
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PI3Kα-IN-1,2100855-80-7
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