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- 保存条件：
Powder: -20°C, 3 years; 4°C, 2 years.In solvent: -80°C, 6 months; -20°C, 1 month.
- 库存：
货期：1-2天
- 供应商：
MedChemExpress LLC
- CAS号：
1256776-89-2
- 规格：
10 mM * 1 mL///1 mg
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FSHR agonist 1
CAS No. : 1256776-89-2
MCE 国际站：FSHR agonist 1
产品活性：FSHR agonist 1 是一种高亲和力和变构卵泡刺激素 (FSH) 受体 (FSHR) 激动剂，pEC50 为 7.72。FSHR agonist 1 与 TMD 形成广泛的相互作用以直接激活 FSHR。
研究领域：Vitamin D Related/Nuclear Receptor
作用靶点：Estrogen Receptor/ERR
In Vitro: The binding of FSHR agonist 1 (compound 21f) to the FSHR TMD pocket induces inward movements of TM6 and TM7, which directly results in FSHR activation.
FSHR agonist 1 (compound 21f) can activate FSHR, LHCGR and TSHR with highly potency and efficacy, while the activation potency for FSHR is more than 10-fold higher than LHCGR (pEC50 of 6.26) and TSHR (pEC50 of 6.48).
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文献和实验Saturation Assays of Radioligand Binding to Receptors and Their Allosteric Modulatory Sites
. The binding of ligands (e.g., the agonist muscimol and antagonist bicuculline) to the GABA receptor requires both α and β subunits. Similarly, both α and γ subunits are required for optimal binding of the agonist diazepam and the antagonist flumazenil
Visualization of Kinase Activity with FRET‐Based Activity Biosensors
transfer to visualize cellular dynamics. In Methods in Cell Biology, Vol. 89: Biophysical Tools for Biologists, Volume 2 (J.J Correia and H.W. Detrich III, eds.) pp. 37‐57. Academic Press, Cambridge, Mass.
Characterization of Dopamine Receptors
Akunne, H.C., Towers, P., Ellis, G.J., Dijkstra, D., Wikstrom, H., Heffner, T.G., Wise, L.D., and Pugsley, T.A. 1995. Characterization of binding of [3H]PD 128907, a selective dopamine D3 receptor agonist
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