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VUF 5681 dihydr
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Please store the product under the recommended conditions in the Certificate of Analysis.
货期:电询
MedChemExpress LLC
639089-06-8
电询
MCE 的所有产品仅用作科学研究或药证申报,我们不为任何个人用途提供产品和服务。
CAS No. : 639089-06-8
MCE 国际站:VUF 5681 dihydrobromide
产品活性:VUF 5681 dihydrobromide 是组胺 H3 receptor 的中性拮抗剂。VUF 5681 dihydrobromide 对组胺 H3 receptor 有部分激动剂的功能。VUF 5681 dihydrobromide 阻断 Thioperamide (HY-12206) 的作用。VUF 5681 dihydrobromide 可用于中枢神经系统疾病的研究。
研究领域:GPCR/G Protein | Neuronal Signaling | Immunology/Inflammation
作用靶点:Histamine Receptor
In Vitro: VUF 5681 dihydrobromide (10 μM) blocks the stimulation of thioperamide in brain tissue.VUF 5681 dihydrobromide (100 nM) inhibits other agonists in CHO-H3-SPAP cells.
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