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- 详细信息
- 文献和实验
- 技术资料
- 保存条件:
Powder: -20°C, 3 years; 4°C, 2 years.In solvent: -80°C, 6 months; -20°C, 1 month.
- 库存:
货期:1-2天
- 供应商:
MedChemExpress LLC
- CAS号:
885104-09-6
- 规格:
10 mM * 1 mL/1 mg/5 mg/10 mg/25 mg
| 规格: | 10 mM * 1 mL | 产品价格: | ¥1447.0 |
|---|---|---|---|
| 规格: | 1 mg | 产品价格: | ¥621.0 |
| 规格: | 5 mg | 产品价格: | ¥1500.0 |
| 规格: | 10 mg | 产品价格: | ¥2400.0 |
| 规格: | 25 mg | 产品价格: | ¥4113.0 |
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LY2389575 hydrochloride
CAS No. : 885104-09-6
MCE 国际站:LY2389575 hydrochloride
产品活性:LY2389575 hydrochloride 是一种选择性和非竞争性的 mGlu3 负变构调节剂 (NAM),IC50 值为 190 nM。LY2389575 hydrochloride 能诱导 Mrc1 水平升高。LY2389575 hydrochloride 还能放大 β 淀粉样蛋白 (Aβ) 的毒性,可用于阿尔兹海默症的研究。
研究领域:GPCR/G Protein | Neuronal Signaling
作用靶点:mGluR
In Vitro: LY2389575 hydrochloride (5 μM; 1 h) induces an increase in Mrc1 levels in microglial cells.
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文献和实验6rKalFCejZJBuWGih0Ooa55R4b1ma5CxEVsQyLeJNULYJQUZ7rZBRYjTJaZFQiLMyFKlNys+J6KKZrop0N0ToIcvFnPLzlGkn2fDyarVpubzyqZec6NbrKZHxlAh/vwhwToU09YIg0q106VyrS5KCoKdVx7Q03tIENxsZy6kM8XQJKQ0zaVRStpF37bu4PTxeG39F2hPxVbeBHZ1NApXYHZowc4UBar37QtyLCLwOBCJJfh3gxaQRgYhARCAiEBF4JQKJeYB0vNK
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