WNK1-IN-1,324022-39-1

MCE 的所有产品仅用作科学研究或药证申报，我们不为任何个人用途提供产品和服务。

WNK1-IN-1

CAS No. : 324022-39-1

MCE 国际站：WNK1-IN-1

产品活性：WNK1-IN-1 是 WNK1 的选择性抑制剂，IC₅₀ 值为 1.6 μM。WNK1-IN-1 抑制 OSR1 磷酸化，IC₅₀ 值为 4.3 μM。WNK1-IN-1 可用于血压调节和癌症的研究。

研究领域：Metabolic Enzyme/Protease

作用靶点：Ser/Thr Protease

In Vitro: WNK1-IN-1 (0-1000 μM; 30 min) shows high potency to WNK1 with an IC₅₀ value of 1.6 μM.
WNK1-IN-1 (0.2-12.5 μM; 24 h) inhibits endogenous OSR1 phosphorylation with an IC₅₀ value of 4.3 μM in MDAMB231 breast-cancer cells.
WNK1-IN-1 (0-100 mM) is 10-fold more potent to WNK1 than WNK3 in Kinase-Glo assay.

相关产品：Bioactive Compound Library Plus  |  Metabolism/Protease Compound Library  |  Anti-Cancer Compound Library  |  Anti-Cardiovascular Disease Compound Library  |  Coagulation and Anti-coagulation Compound Library  |  Highly Selective Inhibitors Library  |  Leupeptin hemisulfate  |  Aprotinin  |  AEBSF hydrochloride  |  Camostat mesylate  |  WNK463  |  Proteinase K  |  Bradykinin  |  Nafamostat mesylate  |  PF-06446846 hydrochloride  |  Inclisiran  |  Trypsin  |  WNK-IN-11  |  Benzamidine hydrochloride  |  Evolocumab  |  SBC-115076  |  Chymotrypsin  |  Trypsin Inhibitor, soybean  |  Pep2-8  |  7-Amino-4-methylcoumarin  |  IPR-803  |  Alirocumab  |  Avoralstat  |  R-IMPP  |  Berotralstat dihydrochloride  |  Bococizumab  |  UKI-1  |  UK122  |  BioE-1115  |  PCSK9-IN-12

热门产品线：重组蛋白  |  化合物库  |  天然产物  |  荧光染料  |  PROTAC  |  同位素标记物

Trending products：Recombinant Proteins  |  Bioactive Screening Libraries  |  Natural Products  |  Dye Reagents  |  PROTAC  |  Isotope-Labeled Compounds