公告提醒:爱必信所有产品和服务仅用于科学研究,不用于临床应用及其他用途提供产品和服务(也不为任何个人提供产品和服务)! 试剂描述: 产品名称:[(3S)-5-甲基-3-(4-吗啉基甲基)-2,3-二氢[1,4]恶嗪并[2,3,4-Hi]吲哚-6-基](1-萘基)甲酮甲烷磺酸酯(1:1) 产品别名: CAS号:131543-25-4 英文别名:[(3S)-5-甲基-3-(4-吗啉基甲基)-2,3-二氢[1,4]恶嗪并[2,3,4-Hi]吲哚-6-基](1-萘基)甲酮甲烷磺酸酯(1:1) 分子量:522.6 分子式:C27H26N2O3 • CH3SO3H 纯度:≥98% 外观:见爱必信官网 保存方法:Store at -20℃ 描述:(−)-WIN 55,212-3 is an aminoalkylindole derivative which acts as a competitive neutral antagonist of the human cannabinoid CB2 receptor, blocking both the stimulating action of CP 55,940 (pA2 = 6.1) and the inverse agonism of SR 144528 (Item No. 9000491) (pEC50 = 5.3).1 (−)-WIN 55,212-3 neither antagonizes nor mimics the effects of Δ9-THC on rat cerebellar membranes, which presumably express the CB1 receptor.2,3 (−)-WIN 55,212-3 also weakly antagonizes the melatonin MT1 and muscarinic M4 receptors but has no effect on several other G protein-coupled receptors.1 应用: 产品信息订购:
产品货号 |
产品名称 |
规格 |
价格 |
大包装及货期 |
abs47044940 |
[(3S)-5-甲基-3-(4-吗啉基甲基)-2,3-二氢[1,4]恶嗪并[2,3,4-Hi]吲哚-6-基](1-萘基)甲酮甲烷磺酸酯(1:1) |
10mg |
2038.00 |
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