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- 详细信息
- 文献和实验
- 技术资料
- 保存条件:
Store at -20℃ for one year(Powder);Store at 2-4℃ for two weeks;Store at -20℃ for six months after dissolution.
- 库存:
99
- 供应商:
爱必信(上海)生物科技有限公司
- CAS号:
152946-68-4
- 规格:
50mg/25mg/10mg/5mg
| 规格: | 50mg | 产品价格: | ¥5943.0 |
|---|---|---|---|
| 规格: | 25mg | 产品价格: | ¥3969.0 |
| 规格: | 10mg | 产品价格: | ¥1577.0 |
| 规格: | 5mg | 产品价格: | ¥1031.0 |
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抑制剂描述: 产品名称:AG-337;Nolatrexed dihydrochloride 产品别名:见爱必信官网 英文别名:AG-337;Nolatrexed dihydrochloride 靶点:Thymidylate synthase CAS:152946-68-4 纯度:98% 外观:见爱必信官网 保存方法:Store at -20℃ for one year(Powder);Store at 2-4℃ for two weeks;Store at -20℃ for six months after dissolution. 描述: Nolatrexed Dihydrochloride is the dihydrochloride salt of nolatrexed, a water-soluble lipophilic quinazoline folate analog with antineoplastic activity. Nolatrexed occupies the folate binding site of thymidylate synthase, resulting in inhibition of thymidylate synthase activity and thymine nucleotide synthesis with subsequent inhibition of DNA replication, DNA damage, S-phase cell cycle arrest, and caspase-dependent apoptosis. This agent also exhibits radiosensitizing activity. 溶解性:DMSO > 10 mM 体外研究: 体内研究:
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文献和实验5’ TCTCACCTCCCAACTGCTTC 3’ AGAGGTTCCTGTCGAGCCGTTTCA 337 IL-5 5’ ATGAGGATGCTTCTGCATTTG 3’ TCAACTTTCTATTATCCACTCGGTGTTCATTAC
Dynamic Monitoring of Cellular Remodeling Induced by the Transforming Growth Factor-β1
by cytochalasin B (CB), Helminthosporium dematioideum (Calbiochem) dissolved in methanol (MeOH). The cells were pretreated with TGF-β1 (10 ng/ml) for 68 h and treated with CB (10 μg/ml) for another 3 h. The cells were monitored continually every 15 s after the CB
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