- ￥788 - 5630
- TargetMol
- 美国
- T37810
- 2025年07月15日
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- 详细信息
- 技术资料
- 保存条件：
零下80~20°C
- 保质期：
Powder: -20°C for 3 years In solvent: -80°C for 2 years
- 英文名：
6',7'-Epoxybergamottin
- 库存：
10
- 供应商：
TargetMol
- CAS号：
206978-14-5
- 规格：
1 mg/5 mg/10 mg
| 规格： | 1 mg | 产品价格： | ￥788.0 |
|---|---|---|---|
| 规格： | 5 mg | 产品价格： | ￥2960.0 |
| 规格： | 10 mg | 产品价格： | ￥5630.0 |
Product Introduction
Bioactivity
英文名:6',7'-Epoxybergamottin
描述:6'7'-Epoxybergamottin is a furanocoumarin found in grapefruit. It is a potent inhibitor of the cytochrome P450 (CYP) isoform CYP3A4 with an IC50 value of 0.30 ppm in a cell-free assay, 0.33 μM in HL7 human liver cells, and 0.22 μM in S9 human intestine cells. It has been studied in the context of drug interactions with grapefruit constituents. It is found in grapefruit juice at concentrations of 0.1-7.4 μM and inhibits the transport of talinolol , a permeability glycoprotein (P-gp/ABCB1) transporter substrate, across Caco-2 cell monolayers (IC50 = 0.7 μM). 6'7'-Epoxybergamottin also has insecticidal properties with a concentration of 5 μg/cm2 leading to 100% mortality of adult olive fruit flies.
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