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4°C, protect from light
- 库存:
货期:1-2天
- 供应商:
MedChemExpress LLC
- CAS号:
309951-18-6
- 规格:
1 mg/5 mg/10 mg/25 mg/50 mg
| 规格: | 1 mg | 产品价格: | ¥304.0 |
|---|---|---|---|
| 规格: | 5 mg | 产品价格: | ¥800.0 |
| 规格: | 10 mg | 产品价格: | ¥1300.0 |
| 规格: | 25 mg | 产品价格: | ¥2500.0 |
| 规格: | 50 mg | 产品价格: | ¥4000.0 |
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BRD4 Inhibitor-24
CAS No. : 309951-18-6
MCE 国际站:BRD4 Inhibitor-24
产品活性:BRD4 Inhibitor-24 (compound 3U) 是一种有效的 BRD4 抑制剂,BRD4 Inhibitor-24 对 MCF7 和 K652 细胞表现出抗肿瘤活性,IC50 分别为 33.7 和 45.9 μM (来自专利 CN107721975A)。
研究领域:Epigenetics
作用靶点:Epigenetic Reader Domain
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科学技术学院田见晖教授团队青年拔尖人才安磊教授题为《BRD4 介导的少量 X 染色体连锁基因转录激活参与早期胚胎 X 染色体剂量上调》(A small proportion of X-linked genes contribute to X chromosome upregulation in early embryos via BRD4-mediated transcriptional activation)的研究论文,揭示了早期胚胎 X 染色体通过上调基因表达,进而平衡性染色体与常染色体剂量的新机
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