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KCC009
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4°C, protect from light
货期:1-2天
MedChemExpress LLC
1 mg/5 mg/10 mg/25 mg
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CAS No. : 744198-19-4
MCE 国际站:KCC009
产品活性:KCC009 是转谷氨酰胺酶 2 的抑制剂,可诱导 p53 途径依赖的放疗敏感性。
研究领域:Metabolic Enzyme/Protease
作用靶点:Glutaminase
In Vitro: The inhibition rates were 15.33±1.46 (%) for H1299/WT-p53 cells, and 14.31±1.90 (%) for H1299/M175H-p53 cells when cells were treated with KCC009 at concentration of 3.91 uM.
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