SSTR5 antagonist 2,2988224-31-

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SSTR5 antagonist 2 hydrochloride

CAS No. :

MCE 国际站：SSTR5 antagonist 2 hydrochloride

产品活性：SSTR5 antagonist 2 hydrochloride (compound 10) 是强效的、具有口服活性的生长激素抑制激素(受体)亚型 5 (SSTR5) 的选择性拮抗剂，有潜力用于 2 型糖尿病的研究。

研究领域：GPCR/G Protein  |  Neuronal Signaling

作用靶点：Somatostatin Receptor

In Vivo: SSTR5 antagonist 2 (compound 10) (10 mg/kg, orally) hydrochloride increases both total and active circulating incretin hormone GLP1 levels in mice at a dose of 10 mg/kg.
SSTR5 antagonist 2 hydrochloride increases pancreatic insulin secretion as well as total and active GLP1 release, and demonstrates synergistic effects in combination with DPP4 inhibitors.

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