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- 详细信息
- 技术资料
- 保存条件:
Powder: -20°C, 3 years; 4°C, 2 years.In solvent: -80°C, 6 months; -20°C, 1 month.
- 库存:
货期:1-2天
- 供应商:
MedChemExpress LLC
- CAS号:
674359-73-0
- 规格:
10 mM * 1 mL/1 mg/5 mg/10 mg/25 mg
| 规格: | 10 mM * 1 mL | 产品价格: | ¥1394.0 |
|---|---|---|---|
| 规格: | 1 mg | 产品价格: | ¥571.0 |
| 规格: | 5 mg | 产品价格: | ¥1488.0 |
| 规格: | 10 mg | 产品价格: | ¥2400.0 |
| 规格: | 25 mg | 产品价格: | ¥4350.0 |
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Rasarfin
CAS No. : 674359-73-0
MCE 国际站:Rasarfin
产品活性:Rasarfin 是 Ras 和 ARF6 的双抑制剂。
研究领域:GPCR/G Protein
作用靶点:Ras
In Vitro: Rasarfin potently inhibits agonist-induced ERK1/2 signaling by GPCRs, and MAPK and Akt signaling by EGFR, as well as prevents cancer cell proliferation.
?Rasarfin blocks GPCR internalization through inhibition of ARF6.
?Rasarfin treatment results in a dose-dependent reduction in MDA-MB-231 cells.
?Rasarfin inhibits the recruitment of the clathrin adaptor AP-2 to β-arrestin2 and receptor internalization, both processes that require active ARF6.
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