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- 详细信息
- 技术资料
- 保存条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
- 库存:
货期:询盘
- 供应商:
MedChemExpress LLC
- CAS号:
851528-10-4
- 规格:
2.5 mg
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Lidocaine-d10 N-Oxide
CAS No. : 851528-10-4
MCE 国际站:Lidocaine-d10 N-Oxide
产品活性:N-Oxide Lidocaine-d10 是 Lidocaine 的氘代物。Lidocaine (Lignocaine) 抑制涉及复杂电压和依赖性的钠通道 (sodium channels)。Lidocaine 通过调节 miR-145 表达和进一步抑制 MEK/ERK 和 NF-κB 信号通路来减少胃癌细胞的生长,迁移和侵袭。Lidocaine 是一种酰胺衍生物,可用于研究室性心律失常。
研究领域:Membrane Transporter/Ion Channel | Stem Cell/Wnt | MAPK/ERK Pathway | NF-κB | Apoptosis
作用靶点:Sodium Channel | MEK | ERK | NF-κB | Apoptosis
In Vitro: Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs.
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