SW155246 is an inhibitor of DNA methyltransferase 1 (DNMT1; IC50 = 1.2 μM).{42214} It is selective for human DNMT1 over murine DNMT3 (IC50 = 38 μM). SW155246 inhibits HeLa and A549 tumor cell growth in a redox-independent manner (IC50s = 8-20 μM). It al
库存:
1 mg, 10 mg, 25 mg, 5 mg
供应商:
Cayman
CAS号:
420092-79-1
A DNMT1 inhibitor (IC50 = 1.2 μM); selective for human DNMT1 over murine DNMT3 (IC50 = 38 μM); inhibits HeLa and A549 tumor cell growth in a redox-independent manner (IC50s = 8-20 μM); inhibits genomic methylation in HeLa cells from 10 to 18.6 μM