Opicapone is a peripherally selective inhibitor of catechol-O-methyltransferase (COMT).{62240} It inhibits COMT activity in rat liver, but not brain, homogenates (ED50 = 1.05 mg/kg). Opicapone (3 mg/kg) increases plasma levels of L-DOPA (Item No. 13248)
英文名:
BIA 9-1067
库存:
1 mg, 10 mg, 5 mg
供应商:
Cayman
CAS号:
923287-50-7
A COMT inhibitor; inhibits COMT activity in rat liver, but not brain, homogenates (ED50 = 1.05 mg/kg); increases L-DOPA plasma levels and reduces 3-OMD plasma levels when administered in combination with benserazide and L-DOPA at 3 mg/kg