Exendin-3 (9-39) amide is a truncated form of the exendin-4 (Item No. 11096) peptide that acts as a potent competitive antagonist for the glucagon-like peptide 1 receptor (GLP-1R; Kd = 1.7 nM in CHL cells transfected with cloned human GLP-1).{27504} It
英文名:
Exendin (9-39)
库存:
1 mg, 500 µg
供应商:
Cayman
CAS号:
133514-43-9
规格:
This biochemical is available in the following size(s) 10 mg, 25 mg, 5 mg - Please inquire
A potent antagonist of GLP-1R (Kd = 1.7 nM); inhibits exendin-3-induced increases in cAMP levels (IC50 = 20 nM); reverses GLP-1 inhibition of feeding behavior in rats when administered at 10 and 100 µg, i.c.v. into the hypothalamus