Peroxisome proliferator-activated receptor γ (PPARγ) is a nuclear receptor with key roles in adipocyte differentiation and glucose homeostasis.{18294,14553} G3335 is a cell-permeable dipeptide that potently antagonizes PPARγ (Kd = 8.34 µM).{28551} It rev
库存:
10 mg, 100 mg, 25 mg, 50 mg
供应商:
Cayman
CAS号:
36099-95-3
规格:
This biochemical is available in the following size(s) 1 mg, 10 mg, 5 mg - Please inquire
A cell-permeable dipeptide that potently antagonizes PPARγ (Kd = 8.34 µM); reversibly and competitively blocks activation of PPARγ by rosiglitazone (IC50 = 8-32 µM); active in vivo, abolishing the protective effects of rosiglitazone in experimental spinal cord injury in rats