Phosphatidylinositol-4-phosphate 5-kinase type-1 γ (PIP5K1C) is a lipid kinase that generates phosphatidylinositol-4,5-bisphosphate (PIP2) in nociceptive dorsal root ganglia (DRG).{26548} Pain sensitization is regulated by multiple signaling pathways tha
库存:
1 mg, 10 mg, 5 mg, 50 mg
供应商:
Cayman
CAS号:
1031602-63-7
规格:
This biochemical is available in the following size(s) 100 µg, 5 mg, 500 µg - Please inquire
A selective, small molecule inhibitor of PIP5K1C (IC50 = 41 nM, Kd = 51 nM); decreases PIP2 membrane levels in cultured DRG neurons by 45%, significantly reducing calcium signaling; displays antinociceptive effects in mouse models of chronic pain