CAY10739 is a soft-drug agonist of the sphingosine-1-phosphate receptor 1 (S1P1; IC50 = 25.12 nM in a β-arrestin recruitment assay) that was designed to prevent systemic effects following topical application.{35828} It is selective for S1P1 over S1P2,
库存:
10 mg, 25 mg, 5 mg, 50 mg
供应商:
Cayman
CAS号:
2328109-05-1
A soft-drug agonist of S1P1 (IC50 = 25.12 nM); selective for S1P1 over S1P2, S1P3, and S1P4 (IC50s = 1,000, >10,000, >10,000 nM, respectively); designed to be activated in the skin and rapidly metabolized to avoid systemic effects