Tilfrinib is an inhibitor of breast tumor kinase/protein tyrosine kinase 6 (BRK/PTK6; IC50 = 3.15 nM).{42337,42338} It is selective for BRK/PTK6 over HER2 (IC50 = 1,300 nM).{42338} Tilfrinib inhibits the growth of MCF-7, HS-578/T, and BT-549 breast canc
库存:
1 mg, 10 mg, 25 mg, 5 mg
供应商:
Cayman
CAS号:
1600515-49-8
规格:
This biochemical is available in the following size(s) 10 mg, 25 mg, 5 mg - Please inquire
An inhibitor of BRK/PTK6 (IC50 = 3.15 nM); selective for BRK/PTK6 over HER2 (IC50 = 1,300 nM); inhibits the growth of MCF-7, HS-578/T, and BT-549 breast cancer cells in vitro (GI50s = 0.99, 1.02, and 1.58 μM, respectively)