CTX-0294885 is a broad spectrum kinase inhibitor that inhibited FAK, FLT3, JAK2, JAK3, Src, Aurora kinase A, and VEGF receptor 3 (IC50s = 4, 1, 3, 28, 2, 18, and 3 nM, respectively) in an initial screen.{40275} In an affinity purification experiment, CT
库存:
1 mg, 10 mg, 25 mg, 5 mg
供应商:
Cayman
CAS号:
1439934-41-4
规格:
This biochemical is available in the following size(s) 1 g, 5 g, 500 mg - Please inquire
A broad spectrum kinase inhibitor used in proteomics; inhibits FAK, Flt3, JAK2, JAK3, Src, Aurora kinase A, and VEGF receptor 3 (IC50s = 4, 1, 3, 28, 2, 18, and 3 nM, respectively); binds to kinases from every major group and captures all members of the AKT family of proteins; captured 235 kinases from MDA-MB-231 breast cancer cells using large-scale kinome profiling